Index 615
1-(4-fl uorophenyl)-3(R)-[3-(4-fl uorophenyl)-
3(S)-hydroxypropyl]-4(S)-(4-
hydroxyphenyl)-2-azetidinone (ezetimibe)
542
4-fl uoro-phenylglycine 481
[S-[R*,S*-(E)]]-7-[4-(4-fl uorophenyl)-5-
(methoxymethyl)-2,6-bis(1-methylethyl)-
3-pyridinyl]-3,5-dihydroxy-6-heptenoate,
sodium salt (cerivastatin sodium) 532
(E,3R,5R)-7-[4-(4-fl uorophenyl)-2-
(methylmethylsulfonyl-amino)-6-propan-
2-yl-pyrimidin-5-yl]-3,5-dihydroxy-hept-
6-enoate, calcium salt (rosuvastatin
calcium) 574
1-(4-fl uorophenyl)-4-(4-methyl-1-
piperidyl)butan-1-one (melperone) 564
3-[1-[4-(4-fl uorophenyl)-4-oxobutyl]-3,6-
dihydro-2H-pyridin-4-yl]-3H-
benzoimidazol-2-one (droperidol) 540
(E,3S,5R)-7-[3-(4-fl uorophenyl)-1-propan-2-yl-
indol-2-yl]-3,5-dihydroxyhept-6-enoate,
sodium salt (fl uvastatin sodium) 554
1-(4-fl uorophenyl)-4-(4-pyridin-2-ylpiperazin-
1-yl)butan-1-one (azaperone) 586
α-fl uoro-α-phenylsulfi nylacetate 264
4-(2-fl uorophenyl)-1,3,8-trimethyl-6H-
pyrazolo[4,5-f][1,4]diazepin-7-one
hydrochloride (zolazepam hydrochloride)
602
α-fl uoro-α-phosphonoacetate 259, 260
Fluoroplex (5-fl uorouracil) 507–12, 548
4(R)-fl uoroproline (Flp)/4(S)-fl uoroproline (fl p)
14, 219, 427–8
2-(fl uoro-propan-2-yloxyphosphoryl)
oxypropane (isofl urophate) 560
[
18
F]fl uoropropyldihydrotetrabenazine (FP-
DTBZ) 366–8
5-fl uoro-2,4(1H,3H)-pyrimdinedione (5-
fl uorouracil) 507–12, 548
fl uoroquinolones 308
fl uorosulfonyldifl uoroacetate (TFDA) 321, 324
9-fl uoro-11,16,17-trihydroxy-17-(2-
hydroxyacetyl)-10,13-dimethyl-6,7,8,9,10,
11,12,13,14,15,16,17-
dodecahydrocyclopenta[a]phenanthren-3-
one (triamcinolone) 600
9-fl uoro-11β,17,21-trihydroxy-16α-
methylpregna-1,4-diene-3,20-dione
(dexamethasone) 538, 588
9-fl uoro-11β,17,21-trihydroxy-16β-
methylpregna-1,4-diene-3,20-dione 17
valerate (betamethasone valerate) 530,
586
α-fl uoro-α-trimethylsilyl acetate 260
fl uorotryptophan 248, 483
5-fl uorouracil (5-FU) 507–12, 548
fl uorous affi nity separation of peptides 413–15
fl uorous biphasic catalysis 412
fl uorous mixture synthesis (FMS) 336–7,
355–6
examples of 339–55
tags (protecting groups) 337–9, 346, 351
fl uorous small-molecule microarrays 415–16
fl uorous tags
in FMS 337–9, 346, 351
in SPPS 413–15
Fluosim (fl umethasone/fl umethasone acetate)
592
Fluothane (halothane) 560, 596
fl uoxetine 512, 513
fl uoxetine hydrochloride (Prozac/Reconcile)
548, 594
fl uoxymesterone (Halotestin) 548
fl uphenazine decanoate 550
fl uphenazine enanthate (Prolixin Enanthate)
550
fl uphenazine hydrochloride 550
fl uprednisolone (Alphadrol) 550
fl uprostenol sodium (Equimate) 52, 594
fl urandrenolide (Cordran) 550
fl urazepam hydrochloride 552
fl urbiprofen (Ansaid) 552
fl urbiprofen sodium (Ocufen) 552
fl urogestone acetate (Synchro-Mate) 596
fl utamide 552
fl uticasone furoate (Flonase) 552
fl uticasone propionate (Advair) 4, 8, 552
fl uvastatin sodium (Lescol) 554
fl uvoxamine maleate 554
FML (fl uorometholone) 548
FMS see fl uorous mixture synthesis
forane (isofl uorane) 560
FP23 peptide (of gp41) 486–7
FS Shampoo (fl uocinolone acetonide) 546
5-FU (5-fl uorouracil) 507–12, 548
Fudr (fl oxuridine) 542
fulvestrant (Faslodex) 554
fusogenic peptides 466, 486–7
GABA (γ-aminobutanoic acid)
aminotransferase 222
GABA (γ-aminobutyric acid) receptor 424
Garner’s aldehyde 220, 241
gatifl oxacin (Zymar) 554
gauche effect 13–16, 190, 427–8
GBC (betamethasone valerate) 586
GCN4 coiled-coil dimer 405–6, 430–1, 432
gefi tinib (Iressa) 554
gelatinase B (MMP-9) 107
gemcitabine hydrochloride (Gemzar) 554